Novel direct C–H borylations of 7-deazapurines to position 8 by B2pin2 under Ir catalysis were followed by Suzuki cross-couplings with aryl halides and other functional group transformations to give diverse 8-substituted 7-deazaadenines.
![Graphical abstract: Direct C–H borylation and C–H arylation of pyrrolo[2,3-d]pyrimidines: synthesis of 6,8-disubstituted 7-deazapurines](/en/Image/Get?imageInfo.ImageType=GA&imageInfo.ImageIdentifier.ManuscriptID=B900218A&imageInfo.ImageIdentifier.Year=2009)
M. Klečka, R. Pohl, B. Klepetářová and M. Hocek, Org. Biomol. Chem., 2009, 7, 866 DOI: 10.1039/B900218A
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