Issue 46, 2010
From the journal:

Chemical Communications

A borylative cyclisation towards indole boronic esters†

Jianhui Huang,a   Simon J. F. Macdonaldb  and  Joseph P. A. Harrity*a  

* Corresponding authors

a Department of Chemistry, University of Sheffield, Sheffield, UK
E-mail: j.harrity@sheffield.ac.uk

b GlaxoSmithKline, Stevenage, Hertfordshire, UK

Abstract

2-Alkynylaniline borylative cyclisations provide a direct means to access indole 3-boronic esters from simple precursors. The Pd-catalysed cyclisation can be merged with cross-coupling processes in the same reaction vessel, moreover, the products can be exploited in C–N bond forming reactions.

Graphical abstract: A borylative cyclisation towards indole boronic esters

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Article information

DOI
https://doi.org/10.1039/C0CC03577G
Article type
Communication
Submitted
31 Aug 2010
Accepted
28 Sep 2010
First published
20 Oct 2010

Chem. Commun., 2010,46, 8770-8772

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A borylative cyclisation towards indole boronic esters

J. Huang, S. J. F. Macdonald and J. P. A. Harrity, Chem. Commun., 2010, 46, 8770 DOI: 10.1039/C0CC03577G

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