Issue 6, 2011
From the journal:

Organic & Biomolecular Chemistry

One-pot double functionalisation of π-deficient heterocyclic lithium reagents†

Anthony Chartoire,a   Corinne Comoya  and  Yves Fort*a  

* Corresponding authors

a Groupe Synthèse Organométallique et Réactivité, SRSMC, Nancy-Université, CNRS, B.P.239, Boulevard des Aiguillettes, Vandoeuvre-Les-Nancy, France
E-mail: Yves.Fort@srsmc.uhp-nancy.fr
Fax: +33 (0)3 83 68 47 85
Tel: +33 (0)3 83 68 47 81

Abstract

Herein, we report an efficient method for the double functionalisation of lithiated halogenopyridines, -pyrazines or -furopyridines through a convenient one-pot electrophilic trapping/nucleophilic substitution sequence.

Graphical abstract: One-pot double functionalisation of π-deficient heterocyclic lithium reagents

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/C0OB00734J
Article type
Paper
Submitted
17 Sep 2010
Accepted
09 Dec 2010
First published
26 Jan 2011

Org. Biomol. Chem., 2011,9, 1839-1845

Permissions

Request permissions

One-pot double functionalisation of π-deficient heterocyclic lithium reagents

A. Chartoire, C. Comoy and Y. Fort, Org. Biomol. Chem., 2011, 9, 1839 DOI: 10.1039/C0OB00734J

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements