Issue 4, 2014

Synthesis of dihydrobenzo[b]furans by diastereoselective acyloxyarylation

Abstract

A highly diastereoselective synthesis of 2-aryl-3-acyloxy-2,3-dihydrobenzofurans by palladium-catalyzed acyloxyarylation involving dearomatization of benzofurans with arylboronic acids and carboxylic acids occurring under mild conditions has been developed.

Graphical abstract: Synthesis of dihydrobenzo[b]furans by diastereoselective acyloxyarylation

Supplementary files

Article information

Article type
Communication
Submitted
26 Sep 2013
Accepted
30 Oct 2013
First published
31 Oct 2013

Chem. Commun., 2014,50, 463-465

Synthesis of dihydrobenzo[b]furans by diastereoselective acyloxyarylation

K. Hata, Z. He, C. G. Daniliuc, K. Itami and A. Studer, Chem. Commun., 2014, 50, 463 DOI: 10.1039/C3CC47350C

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