Issue 21, 2014
From the journal:

Chemical Communications

Copper-catalyzed ortho-C–H amination of protected anilines with secondary amines†

Ángel Manu Martínez,a   Nuria Rodríguez,*a   Ramón Gómez Arrayás*a  and  Juan C. Carreteroa  

* Corresponding authors

a Departamento de Química Orgánica, Universidad Autónoma de Madrid, Cantoblanco, 28049 Madrid, Spain
E-mail: n.rodriguez@uam.es, ramon.gomez@uam.es

Abstract

A practical Cu-catalyzed picolinamide-directed o-amination of anilines showing excellent mono-substitution selectivity and high functional group tolerance has been developed.

Graphical abstract: Copper-catalyzed ortho-C–H amination of protected anilines with secondary amines

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Article information

DOI
https://doi.org/10.1039/C3CC49633C
Article type
Communication
Submitted
19 Dec 2013
Accepted
22 Jan 2014
First published
03 Feb 2014

Chem. Commun., 2014,50, 2801-2803

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Copper-catalyzed ortho-C–H amination of protected anilines with secondary amines

Á. M. Martínez, N. Rodríguez, R. G. Arrayás and J. C. Carretero, Chem. Commun., 2014, 50, 2801 DOI: 10.1039/C3CC49633C

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