Issue 26, 2014
From the journal:

Organic & Biomolecular Chemistry

Synthesis of 2-C-substituted benzothiazoles via a copper-promoted domino condensation/S-arylation/heterocyclization process†

Haoyue Xiang,‡ab   Jin Qi,‡a   Qian He,b   Min Jiang,*a   Chunhao Yang*b  and  Lianfu Denga  

* Corresponding authors

a Shanghai Key Laboratory for Bone and Joint Diseases, Shanghai Institute of Traumatology and Orthopaedics, Shanghai Ruijin Hospital, Shanghai Jiaotong University School of Medicine, Shanghai, China
E-mail: jiangm263@163.com

b State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai, P.R. China
E-mail: chyang@simm.ac.cn
Fax: +86-21-50806770
Tel: +86-21-50806770

Abstract

Two series of extremely useful 2-C-substituted benzothiazoles containing gem-bisphosphonates and aryl-substituted nitriles were synthesized here via a copper-promoted domino condensation/S-arylation/heterocyclization process.

Graphical abstract: Synthesis of 2-C-substituted benzothiazoles via a copper-promoted domino condensation/S-arylation/heterocyclization process

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Article information

DOI
https://doi.org/10.1039/C4OB00564C
Article type
Paper
Submitted
14 Mar 2014
Accepted
01 May 2014
First published
01 May 2014

Org. Biomol. Chem., 2014,12, 4633-4636

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Synthesis of 2-C-substituted benzothiazoles via a copper-promoted domino condensation/S-arylation/heterocyclization process

H. Xiang, J. Qi, Q. He, M. Jiang, C. Yang and L. Deng, Org. Biomol. Chem., 2014, 12, 4633 DOI: 10.1039/C4OB00564C

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