Issue 37, 2016

Double heteroannulation of S,N-acetals: a facile access to quinolone derivatives

Abstract

A rapid construction of quinolone fused heterocycles from single S,N-acetal precursors via double heteroannulation is described. The base, radical and metal-mediated reactions can control the C–N, C–S and C–O bond formations of the S,N-acetal with high chemoselectivity.

Graphical abstract: Double heteroannulation of S,N-acetals: a facile access to quinolone derivatives

Supplementary files

Article information

Article type
Paper
Submitted
22 Jul 2016
Accepted
19 Aug 2016
First published
19 Aug 2016

Org. Biomol. Chem., 2016,14, 8781-8788

Double heteroannulation of S,N-acetals: a facile access to quinolone derivatives

M. Janni, S. Arora and S. Peruncheralathan, Org. Biomol. Chem., 2016, 14, 8781 DOI: 10.1039/C6OB01568A

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