A Suzuki–Miyaura cross-coupling reaction was developed on unprotected ortho-bromoanilines. This operationally simple reaction was developed for the diversification of glucocorticoid receptor modulators (GRMs), showed compatibility to various boronic esters featuring unique functionalities, and was demonstrated on a gram scale.
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A. E. Lubaev, C. C. Marvin, A. W. Dombrowski and Z. Qureshi, RSC Adv., 2024, 14, 29184 DOI: 10.1039/D4RA03725A
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