Issue 6, 2010
From the journal:

Chemical Communications

Efficient synthesis of aminopyridine derivatives by copper catalyzed amination reactions†

Mohammed K. Elmkaddem,a   Cédric Fischmeister,*a   Christophe M. Thomas*b  and  Jean-Luc Renaud*c  

* Corresponding authors

a UMR 6226-CNRS-Université de Rennes 1, Sciences Chimiques de Rennes, Catalyse et Organométalliques, Campus de Beaulieu, avenue du général Leclerc, 35042 Rennes cedex, France
E-mail: cedric.fischmeister@univ-rennes1.fr
Fax: +33(0)223236939
Tel: +33(0)223235998

b ENSCP, UMR CNRS 7223, 11 rue Pierre et Marie Curie, 75005 Paris, France
E-mail: christophe-thomas@enscp.fr
Fax: +33(0)143260061
Tel: +33(0)144276721

c Laboratoire de Chimie Moléculaire et Thioorganique, UMR 6507, INC3M, FR 3038, ENSICAEN-Université de Caen, 14050 Caen, France
E-mail: jean-luc.renaud@ensicaen.fr
Fax: +33(0)231452877
Tel: +33(0)231452842

Abstract

A copper(I) catalyzed amination reaction utilizing aqueous ammonia and operating under mild conditions is presented. This method was employed for the efficient synthesis of various aminopyridine derivatives bearing electron withdrawing and electron donating groups.

Graphical abstract: Efficient synthesis of aminopyridine derivatives by copper catalyzed amination reactions

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Article information

DOI
https://doi.org/10.1039/B916569J
Article type
Communication
Submitted
11 Aug 2009
Accepted
13 Oct 2009
First published
07 Dec 2009

Chem. Commun., 2010,46, 925-927

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Efficient synthesis of aminopyridine derivatives by copper catalyzed amination reactions

M. K. Elmkaddem, C. Fischmeister, C. M. Thomas and J. Renaud, Chem. Commun., 2010, 46, 925 DOI: 10.1039/B916569J

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